PeptideDB

BMS-740808

CAS: 280118-23-2 F: C31H27F3N6O3 W: 588.58

BMS-740808 is a potent, selective and orally active factor Xa inhibitorwith a Ki of 30 pM. BMS-740808 shows >1000-fold f
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This product is for research use only, not for human use. We do not sell to patients.

Bioactivity BMS-740808 is a potent, selective and orally active factor Xa inhibitor with a Ki of 30 pM. BMS-740808 shows >1000-fold for factor Xa than other proteases[1].
CAS 280118-23-2
Formula C31H27F3N6O3
Molar Mass 588.58
Transport Room temperature in continental US; may vary elsewhere.
Storage

Please store the product under the recommended conditions in the Certificate of Analysis.

Reference [1]. Donald J P Pinto, et al. 1-[3-Aminobenzisoxazol-5'-yl]-3-trifluoromethyl-6-[2'-(3-(R)-hydroxy-N-pyrrolidinyl)methyl-[1,1']-biphen-4-yl]-1,4,5,6-tetrahydropyrazolo-[3,4-c]-pyridin-7-one (BMS-740808) a highly potent, selective, efficacious, and orally bioavailable inhibitor of blood coagulation factor Xa. Bioorg Med Chem Lett. 2006 Aug 1;16(15):4141-7.