| Bioactivity | BI-167107 is a high affinity, full agonist that binds to the β2 adrenergic receptor (β2AR) with a dissociation constant Kd of 84 pM[1]. | ||||||||||||
| Target | Kd: 84 pM (β2AR) | ||||||||||||
| Invitro | Compared to other βAR ligands, BI-167107 displays nanomolar affinities and slow off-rates[1]. | ||||||||||||
| Name | BI-167107 | ||||||||||||
| CAS | 1202235-68-4 | ||||||||||||
| Formula | C21H26N2O4 | ||||||||||||
| Molar Mass | 370.44 | ||||||||||||
| Appearance | Solid | ||||||||||||
| Transport | Room temperature in continental US; may vary elsewhere. | ||||||||||||
| Storage |
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| Reference | [1]. Rasmussen SG, et al. Structure of a nanobody-stabilized active state of the β(2) adrenoceptor. Nature. 2011 Jan 13;469(7329):175-80. |