Bioactivity | BET bromodomain inhibitor 3 is BET bromodomain inhibitor. BET bromodomain inhibitor 3 has inhibitory effect against BrdT with Ki value of > 40 µM. BET bromodomain inhibitor 3 can be used for the research of contraception, cancer, and heart disease[1]. |
Target | Ki: > 40 µM (BrdT) |
Invitro | BET bromodomain inhibitor 3 对 BrdT 有抑制作用,Ki 值 > 40 µM[1]。 |
Name | BET bromodomain inhibitor 3 |
CAS | 854137-39-6 |
Formula | C18H17N3O4 |
Molar Mass | 339.35 |
Transport | Room temperature in continental US; may vary elsewhere. |
Storage | Please store the product under the recommended conditions in the Certificate of Analysis. |
Reference | [1]. Ayoub AM, et al. BET Bromodomain Inhibitors with One-Step Synthesis Discovered from Virtual Screen [published correction appears in J Med Chem. 2017 Jul 27;60(14):6458]. J Med Chem. 2017;60(12):4805-4817. |