| Bioactivity | BET-IN-17 (compound 16) is a pan-inhibitor of BET with pIC50s of 7.8 and 7.6 for BET BD1 and BET BD2, respectively[1]. |
| Target | pIC50: 7.8 (BET BD1), 7.6 (BET BD2) |
| Name | BET-IN-17 |
| Formula | C30H36N4O2 |
| Molar Mass | 484.63 |
| Transport | Room temperature in continental US; may vary elsewhere. |
| Storage | Please store the product under the recommended conditions in the Certificate of Analysis. |
| Reference | [1]. Bamborough P, et al. Design and Characterization of 1, 3-Dihydro-2 H-benzo [d] azepin-2-ones as Rule-of-5 Compliant Bivalent BET Inhibitors[J]. ACS Medicinal Chemistry Letters, 2023.. . . |