BET-IN-15

CAS: 2408994-22-7 F: C21H18F2N4O3S W: 444.45

BET-IN-15 (compound 1) is a potent and orally active BET inhibitor with IC50 values of 0.64, 0.25 nM for BRD4-BD1, BRD4-

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Bioactivity	BET-IN-15 (compound 1) is a potent and orally active BET inhibitor with IC50 values of 0.64, 0.25 nM for BRD4-BD1, BRD4-BD2, respectively. BET-IN-15 shows antiproliferative activity[1].
Invitro	BET-IN-15 (compound 1) (72 h) 显示出抗增殖活性，对于 MV4-11、Kasumi-1 细胞的 IC50s 分别为 3.14、1.56 nM[1]。
In Vivo	BET-IN-15 (compound 1) (72 h) 显示出抗增殖活性，对于 MV4-11、Kasumi-1 细胞的IC50s 分别为 3.14、1.56 nM[1]。
Name	BET-IN-15
CAS	2408994-22-7
Formula	C21H18F2N4O3S
Molar Mass	444.45
Transport	Room temperature in continental US; may vary elsewhere.
Storage	Please store the product under the recommended conditions in the Certificate of Analysis.
Reference	[1]. WenWei Xu, et al. Crystal form and salt form of bromine domain protein inhibitor and preparation method therefor. WO2021143922A1.

N-Methyl-DL-valine hydrochloride