| Bioactivity | BET-IN-1 is a potent BET inhibitor that has excellent brain penetration and reasonable metabolic stability. |
| Name | BET-IN-1 |
| Formula | C23H24ClFN4O3S |
| Molar Mass | 490.98 |
| Transport | Room temperature in continental US; may vary elsewhere. |
| Storage | Please store the product under the recommended conditions in the Certificate of Analysis. |
| Reference | [1]. Bai P, et al. Design, Synthesis, and Evaluation of Thienodiazepine Derivatives as Positron Emission Tomography Imaging Probes for Bromodomain and Extra-Terminal Domain Family Proteins. J Med Chem. 2021 Oct 14;64(19):14745-14756. |