| Bioactivity | BChE-IN-5 is a potent and selective BChE inhibitor of hBChE over hAChE with an IC50 of 2.8 nM for BChE. BChE-IN-5 has the potential for the research of alzheimer’s disease[1]. |
| Target | BChE |
| Invitro | BChE-IN-5 (compound 18) shows inhibitory potencies for hBChE and hAChE with IC50s of 2.8 nM, 16000 nM, respectively[1]. |
| Name | BChE-IN-5 |
| Formula | C30H42N4O |
| Molar Mass | 474.68 |
| Transport | Room temperature in continental US; may vary elsewhere. |
| Storage | Please store the product under the recommended conditions in the Certificate of Analysis. |
| Reference | [1]. Meden A, et al. Structure-activity relationship study of tryptophan-based butyrylcholinesterase inhibitors. Eur J Med Chem. 2020 Dec 15;208:112766. |