| Bioactivity | Axelopran (TD-1211) is an antagonist for opioid receptor, with pKi of 9.8, 8.8 and 9.9, for human recombinant μ and δ receptors and guinea pig κ receptors, respectively[1]. |
| CAS | 949904-48-7 |
| Formula | C26H39N3O4 |
| Molar Mass | 457.61 |
| Transport | Room temperature in continental US; may vary elsewhere. |
| Storage | Please store the product under the recommended conditions in the Certificate of Analysis. |
| Reference | [1]. Tsuruda PR, et al., The in vitro pharmacological profile of TD-1211, a neutral opioid receptor antagonist. Naunyn Schmiedebergs Arch Pharmacol. 2013 Jun;386(6):479-91. |