Bioactivity | Aprocitentan (Standard) is the analytical standard of Aprocitentan. This product is intended for research and analytical applications. Aprocitentan (ACT-132577) is the major and pharmacologically active metabolite of Macitentan. Aprocitentan is dual ETA/ETB antagonist with IC50s of 3.4 nM and 987 nM, and pA2 valus of 6.7 and 5.5, respectively. |
CAS | 1103522-45-7 |
Formula | C16H14Br2N6O4S |
Molar Mass | 546.19 |
Storage | Please store the product under the recommended conditions in the Certificate of Analysis. |