PeptideDB

Apalutamide-d4

CAS: 1638885-65-0 F: C21H11D4F4N5O2S W: 481.46

Apalutamide-d4 is a deuterium labeled Apalutamide. Apalutamide is a potent and competitive androgen receptor (AR) antago
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This product is for research use only, not for human use. We do not sell to patients.

Bioactivity Apalutamide-d4 is a deuterium labeled Apalutamide. Apalutamide is a potent and competitive androgen receptor (AR) antagonist, binding AR with an IC50 of 16 nM[1].
Name Apalutamide-d4
CAS 1638885-65-0
Formula C21H11D4F4N5O2S
Molar Mass 481.46
Appearance Solid
Transport Room temperature in continental US; may vary elsewhere.
Storage
Powder -20°C 3 years
4°C 2 years
In solvent -80°C 6 months
-20°C 1 month
Reference [1]. Clegg NJ, et al. ARN-509: a novel antiandrogen for prostate cancer treatment. Cancer Res. 2012 Mar 15;72(6):1494-503.