Antitumor agent-136_product_DataBase

CAS: 2484876-94-8 F: C58H76N10O11S3 W: 1185.48

Antitumor Agent-136 (Compound 17) is a potent broad-spectrum antitumor agent and a NAMPT inhibitor with an IC50 of 9.5 n

This product is for research use only, not for human use. We do not sell to patients.

Bioactivity	Antitumor Agent-136 (Compound 17) is a potent broad-spectrum antitumor agent and a NAMPT inhibitor with an IC50 of 9.5 nM. Antitumor Agent-136 can reduce the levels of intracellular and extracellular NAMPT protein through the ubiquitin proteasome pathway, thus achieving tumor inhibition[1].
Target	IC50: 9. 5 nM (NAMPT).
Name	Antitumor agent-136
CAS	2484876-94-8
Formula	C58H76N10O11S3
Molar Mass	1185.48
Transport	Room temperature in continental US; may vary elsewhere.
Storage	Please store the product under the recommended conditions in the Certificate of Analysis.
Reference	[1]. 盛春泉, et al. NAMPT protein degradation targeting chimera and preparation method and application thereof. China. CN111454327. 2020-07028.

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