| Bioactivity | Androgen receptor antagonist 2 (example 12) is an androgen receptor antagonist. Androgen receptor antagonist 2 can be used for prostate cancer and male hair loss research[1]. | |||||||||
| Invitro | Androgen receptor antagonist 2 (example 12) inhibits PSA production with an IC50 of 0.28 μM in LNCaP cells[1].Androgen receptor antagonist 2 (2.5 μM, 48 h) inhibits prostate cancer cells viability[1]. Cell Viability Assay[1] Cell Line: | |||||||||
| In Vivo | Androgen receptor antagonist 2 (example 12) (0.2% and 1% concentration, 20 mL/mouse; topical application; twice daily for 4 weeks) promotes hair growth in mice[1]. Animal Model: | |||||||||
| Name | Androgen receptor antagonist 2 | |||||||||
| CAS | 1272719-00-2 | |||||||||
| Formula | C21H15F5N4O2S | |||||||||
| Molar Mass | 482.43 | |||||||||
| Appearance | Solid | |||||||||
| Transport | Room temperature in continental US; may vary elsewhere. | |||||||||
| Storage |
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| Reference | [1]. Youzhi Tong. Androgen receptor antagonists and uses thereof. WO2011029392A1. |
Androgen receptor antagonist 2
CAS: 1272719-00-2 F: C21H15F5N4O2S W: 482.43
Androgen receptor antagonist 2 (example 12) is an androgen receptor antagonist. Androgen receptor antagonist 2 can be us
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