Bioactivity | Androgen receptor antagonist 11 (compund N29) is a derivative of the androgen receptor (AR) antagonist M17-B15, and is a selective and orally active AR antagonist (IC50=18 nM).[1]. |
CAS | 2719816-32-5 |
Formula | C20H19F3N4O3S |
Molar Mass | 452.45 |
Transport | Room temperature in continental US; may vary elsewhere. |
Storage | Please store the product under the recommended conditions in the Certificate of Analysis. |
Reference | [1]. Liao J, et al. Discovery of Thiadiazoleamide Derivatives as Potent, Selective, and Orally Available Antagonists Disrupting Androgen Receptor Homodimer. J Med Chem. 2024 Oct 10;67(19):17520-17541. |