| Bioactivity | Androgen receptor-IN-6 (compound 16) is an orally available androgen receptor (Androgen Receptor) potent inhibitor (IC50=0.12 μM in vitro), targeting the disordered N-terminal domain (NTD). Androgen receptor-IN-6 has good Caco2 cell membrane permeability and has an oral activity (F/%) of 16% in male CD-1 mice[1]. |
| Name | Androgen receptor-IN-6 |
| Formula | C16H15N3OS |
| Molar Mass | 297.37 |
| Transport | Room temperature in continental US; may vary elsewhere. |
| Storage | Please store the product under the recommended conditions in the Certificate of Analysis. |
| Reference | [1]. Henry M C et al. Synthesis and evaluation of small molecule inhibitors of the androgen receptor N-terminal domain[J]. ACS Medicinal Chemistry Letters, 2023. |
Androgen receptor-IN-6
CAS: F: C16H15N3OS W: 297.37
Androgen receptor-IN-6 (compound 16) is an orally available androgen receptor (Androgen Receptor) potent inhibitor (IC50
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