Bioactivity | Adenosine receptor antagonist 4 (compound 2) is an adenosine A1 receptor antagonist with a Ki of 101 nM for human A1 receptor[1]. | ||||||||||||
Name | Adenosine receptor antagonist 4 | ||||||||||||
CAS | 133240-06-9 | ||||||||||||
Formula | C10H13N3 | ||||||||||||
Molar Mass | 175.23 | ||||||||||||
Appearance | Solid | ||||||||||||
Transport | Room temperature in continental US; may vary elsewhere. | ||||||||||||
Storage |
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Reference | [1]. Lisa C W Chang, et al. 2,6,8-trisubstituted 1-deazapurines as adenosine receptor antagonists. J Med Chem. 2007 Feb 22;50(4):828-34. |