Bioactivity | Acetalin-3 (Ac-RFMWMT-NH2), a hexapeptide, is a μ opioid receptor antagonist with high affinity for μ and κ3 opioid receptor, weak affinity for κ1 receptors and no affinity for κ2 receptors[1]. |
Name | Acetalin-3 |
CAS | 152274-65-2 |
Sequence | Ac-Arg-Phe-Met-Trp-Met-Thr-NH2 |
Shortening | Ac-RFMWMT-NH2 |
Formula | C42H61N11O8S2 |
Molar Mass | 912.13 |
Transport | Room temperature in continental US; may vary elsewhere. |
Storage | Please store the product under the recommended conditions in the Certificate of Analysis. |
Reference | [1]. C T Dooley, et al. Acetalins: opioid receptor antagonists determined through the use of synthetic peptide combinatorial libraries. Proc Natl Acad Sci U S A. 1993 Nov 15;90(22):10811-5. |