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AS2717638

CAS: 2148339-28-8 F: C25H25N3O5 W: 447.48

AS2717638 is an oral active and selective lysophosphatidic acid receptor 5 (LPA5) antagonist, with an IC50 of 38 nM for
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Bioactivity AS2717638 is an oral active and selective lysophosphatidic acid receptor 5 (LPA5) antagonist, with an IC50 of 38 nM for hLPA5. AS2717638 also significantly improves PGE2-, PGF2α-, and AMPA-induced allodynia[1].
Target IC50: 38 nM (hLPA5).
Name AS2717638
CAS 2148339-28-8
Formula C25H25N3O5
Molar Mass 447.48
Appearance Solid
Transport Room temperature in continental US; may vary elsewhere.
Storage
Powder -20°C 3 years
4°C 2 years
In solvent -80°C 6 months
-20°C 1 month
Reference [1]. Murai N, et al. Analgesic effects of novel lysophosphatidic acid receptor 5 antagonist AS2717638 in rodents. Neuropharmacology. 2017 Nov;126:97-107.

TC-S 7009

Benproperine phosphate

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Is for research use only, not for human use. We do not sell to patients.