Bioactivity | AMPA receptor modulator-2 (Example 134) is a AMPA receptor modulator, with a pIC50 of 10.1 for TARPγ2 dependent AMPA receptor[1]. pIC50 = -lgIC50. | ||||||||||||
Target | pIC50: AMPA receptor (10.1). | ||||||||||||
Name | AMPA receptor modulator-2 | ||||||||||||
CAS | 2034181-36-5 | ||||||||||||
Formula | C15H6F6N4OS | ||||||||||||
Molar Mass | 404.29 | ||||||||||||
Appearance | Solid | ||||||||||||
Transport | Room temperature in continental US; may vary elsewhere. | ||||||||||||
Storage |
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Reference | [1]. BERRY CYNTHIA G B (US), et al. AZABENZIMIDAZOLES AND THEIR USE AS AMPA RECEPTOR MODULATORS. Patent. WO2016176460. |