| Bioactivity | AMG0347 is a transient receptor potential type V1 receptor antagonist. AMG0347 inhibits activation of the rat TRPV1 channel by heat (IC50 = 0.2 nm), protons (IC50= 0.8 nm), or capsaicin (IC50 = 0.7 nm)[1]. |
| Name | AMG0347 |
| CAS | 946615-43-6 |
| Formula | C24H26F3N3O2 |
| Molar Mass | 445.48 |
| Transport | Room temperature in continental US; may vary elsewhere. |
| Storage | Please store the product under the recommended conditions in the Certificate of Analysis. |
| Reference | [1]. Chaoran Wu, et al. Effect of AMG0347, a Transient Receptor Potential Type V1 Receptor Antagonist, and Morphine on Pain Behavior after Plantar Incision。Anesthesiology. 2008 Jun;108(6):1100-8. |
AMG0347
CAS: 946615-43-6 F: C24H26F3N3O2 W: 445.48
AMG0347 is a transient receptor potential type V1 receptor antagonist. AMG0347 inhibits activation of the rat TRPV1 chan
Sales Email：peptidedb@qq.com
This product is for research use only, not for human use. We do not sell to patients.