| Bioactivity | AChE/BChE-IN-8 (Compound 5a) is an uncompetitive AChE and mixed BChE inhibitor with Ki values of 0.788 μM and 2.364 μM against Electrophorus electricus AChE (EeAChE) and equine BChE (eqBChE), respectively. AChE/BChE-IN-8 can cross the BBB and has low cytotoxicity[1]. |
| Target | Ki: 0.788 μM (EeAChE), 2.364 μM (eqBChE) |
| Name | AChE/BChE-IN-8 |
| CAS | 2421120-96-7 |
| Formula | C26H32N2O2 |
| Molar Mass | 404.54 |
| Transport | Room temperature in continental US; may vary elsewhere. |
| Storage | Please store the product under the recommended conditions in the Certificate of Analysis. |
| Reference | [1]. Bortolami M, et al. New deferiprone derivatives as multi-functional cholinesterase inhibitors: design, synthesis and in vitro evaluation. Eur J Med Chem. 2020 Jul 15;198:112350. |
AChE/BChE-IN-8
CAS: 2421120-96-7 F: C26H32N2O2 W: 404.54
AChE/BChE-IN-8 (Compound 5a) is an uncompetitive AChE and mixed BChE inhibitor with Ki values of 0.788 μM and 2.364 μM
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