| Bioactivity | ABCG2-IN-1 (compound K2), a Ko143 analog, is an orally active ABCG2 inhibitor with an IC50 of 0.13 μM. ABCG2-IN-1 has favorable oral pharmacokinetic profiles in mice[1]. |
| Target | IC50: 0.13 μM (ABCG2) |
| Name | ABCG2-IN-1 |
| CAS | 2559759-40-7 |
| Formula | C26H36N4O4 |
| Molar Mass | 468.59 |
| Transport | Room temperature in continental US; may vary elsewhere. |
| Storage | Please store the product under the recommended conditions in the Certificate of Analysis. |
| Reference | [1]. Junjie Zhu, et al. Metabolism-guided development of Ko143 analogs as ABCG2 inhibitors. Eur J Med Chem. 2023 Nov 5;259:115666. |
ABCG2-IN-1
CAS: 2559759-40-7 F: C26H36N4O4 W: 468.59
ABCG2-IN-1 (compound K2), a Ko143 analog, is an orally active ABCG2 inhibitor with an IC50 of 0.13 μM. ABCG2-IN-1 has f
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