Bioactivity | AA10 is a potent and irreversible transglutaminase 2 (TG2) inhibitor for cancer research[1]. |
Name | AA10 |
CAS | 2134106-02-6 |
Formula | C32H36N4O5 |
Molar Mass | 556.65 |
Transport | Room temperature in continental US; may vary elsewhere. |
Storage | Please store the product under the recommended conditions in the Certificate of Analysis. |
Reference | [1]. Akbar A, et al. Structure-Activity Relationships of Potent, Targeted Covalent Inhibitors That Abolish Both the Transamidation and GTP Binding Activities of Human Tissue Transglutaminase. J Med Chem. 2017 Sep 28;60(18):7910-7927. |