| Bioactivity | A71378 is a selectivity CCK-A receptor agonist the IC50 values of 0.4 nM, 300 nM, and 1,200 nM for the pancreatic CCK-A, cortical CCK-B, and gastrin receptor, respectively. A71378 elicits pancreatic amylase secretion (EC50 = 0.16 nM) and ileal muscle contraction (EC50 = 3.7 nM)[1]. |
| CAS | 127902-33-4 |
| Formula | C48H62N8O13S |
| Molar Mass | 991.12 |
| Transport | Room temperature in continental US; may vary elsewhere. |
| Storage | Please store the product under the recommended conditions in the Certificate of Analysis. |
| Reference | [1]. Lin CW, et al. A71378: a CCK agonist with high potency and selectivity for CCK-A receptors. Am J Phy |