| Bioactivity | A2AAR antagonist 1 (compound 21a) is an A2AAR (adenosine A2A receptor) antagonist with a Ki value of 20 nM. A2AAR antagonist 1 shows high ligand efficiency, and it can be used for the research of neurodegenerative diseases[1]. |
| Invitro | A2AAR antagonist 1 (0-10 μM; 1 h) shows a high affinity towards A2AAR with a Ki value of 20 nM[1]. |
| Name | A2AAR antagonist 1 |
| CAS | 1784491-64-0 |
| Formula | C12H8BrN3O |
| Molar Mass | 290.12 |
| Transport | Room temperature in continental US; may vary elsewhere. |
| Storage | Please store the product under the recommended conditions in the Certificate of Analysis. |
| Reference | [1]. Bolteau R, et al. High ligand efficiency quinazoline compounds as novel A2A adenosine receptor antagonists. Eur J Med Chem. 2022 Nov 5;241:114620. |
A2AAR antagonist 1
CAS: 1784491-64-0 F: C12H8BrN3O W: 290.12
A2AAR antagonist 1 (compound 21a) is an A2AAR (adenosine A2A receptor) antagonist with a Ki value of 20 nM. A2AAR antago
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