| Bioactivity | 8-Cyclopentyl-1,3-dimethylxanthine (Compound 2a) is a selective adenosine A1 receptor antagonist with Kis of 10.9 nM and 1440 nM for A1 receptor and A2 receptor, respectively[1]. |
| Target | Ki: 10.9 nM (A1 receptor), 1440 nM (A2 receptor) |
| Name | 8-Cyclopentyl-1,3-dimethylxanthine |
| CAS | 35873-49-5 |
| Formula | C12H16N4O2 |
| Molar Mass | 248.28 |
| Transport | Room temperature in continental US; may vary elsewhere. |
| Storage | Please store the product under the recommended conditions in the Certificate of Analysis. |
| Reference | [1]. K A Jacobson, et al. Sulfur-containing 1,3-dialkylxanthine derivatives as selective antagonists at A1-adenosine receptors. J Med Chem. 1989 Aug;32(8):1873-9. |