PeptideDB

8-Cyclopentyl-1,3-dimethylxanthine

CAS: 35873-49-5 F: C12H16N4O2 W: 248.28

8-Cyclopentyl-1,3-dimethylxanthine (Compound 2a) is a selective adenosine A1 receptor antagonist with Kis of 10.9 nM and
Sales Email:peptidedb@qq.com

This product is for research use only, not for human use. We do not sell to patients.

Bioactivity 8-Cyclopentyl-1,3-dimethylxanthine (Compound 2a) is a selective adenosine A1 receptor antagonist with Kis of 10.9 nM and 1440 nM for A1 receptor and A2 receptor, respectively[1].
Target Ki: 10.9 nM (A1 receptor), 1440 nM (A2 receptor)
Name 8-Cyclopentyl-1,3-dimethylxanthine
CAS 35873-49-5
Formula C12H16N4O2
Molar Mass 248.28
Transport Room temperature in continental US; may vary elsewhere.
Storage

Please store the product under the recommended conditions in the Certificate of Analysis.

Reference [1]. K A Jacobson, et al. Sulfur-containing 1,3-dialkylxanthine derivatives as selective antagonists at A1-adenosine receptors. J Med Chem. 1989 Aug;32(8):1873-9.