| Bioactivity | 6-Methylflavone is an activator of α1β2γ2L and α1β2 GABAA receptors. | ||||||||||||
| Invitro | 6-Methylflavone is an activator of α1β2γ2L and α1β2 GABAA receptors. 6-Methylflavone enhances the normal response to GABA at recombinant α1β2γ2L and α1β2 GABAA receptors (P<0.0001) at concentrations from 1 to 100 μM. 6-Methylflavone (60 μM) shifts the GABA dose-response curve to the left (n=4, F=16.38, P=0.0004), decreasing the mean EC50 at α1β2γ2L GABAA receptors by 33±5.4%[1]. | ||||||||||||
| Name | 6-Methylflavone | ||||||||||||
| CAS | 29976-75-8 | ||||||||||||
| Formula | C16H12O2 | ||||||||||||
| Molar Mass | 236.27 | ||||||||||||
| Transport | Room temperature in continental US; may vary elsewhere. | ||||||||||||
| Storage |
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