Bioactivity | 5-HT6/5-HT2AR antagonist-1 is a potent dual 5-HT6/5-HT2AR antagonist with Ki values of 11 nM and 39 nM, respectively[1]. |
Name | 5-HT6/5-HT2AR antagonist-1 |
Formula | C21H26N6S |
Molar Mass | 394.54 |
Transport | Room temperature in continental US; may vary elsewhere. |
Storage | Please store the product under the recommended conditions in the Certificate of Analysis. |
Reference | [1]. Katarzyna Kucwaj-Brysz, et al. An exit beyond the pharmacophore model for 5-HT 6 R agents - a new strategy to gain dual 5-HT 6/5-HT 2A action for triazine derivatives with procognitive potential. Bioorg Chem. 2022 Apr;121:105695. |