Bioactivity | 22-Hydroxy Mifepristone (RU 42698) is an orally active hydroxylated alcoholic metabolite with antiprogestational and antiglucocorticoidal activities, which contains an Alkyne group and can undergo copper-catalyzed azide-alkyne cycloaddition (CuAAc) with molecules containing Azide groups. The relative binding affinity of 22-Hydroxy Mifepristone to the human glucocorticoid receptor is 48%[1][2]. |
CAS | 105012-15-5 |
Formula | C31H39NO3 |
Molar Mass | 473.65 |
Transport | Room temperature in continental US; may vary elsewhere. |
Storage | Please store the product under the recommended conditions in the Certificate of Analysis. |
Reference | [1]. Lähteenmäki P, et al. Pharmacokinetics and metabolism of RU 486. J Steroid Biochem. 1987;27(4-6):859-63. [2]. Heikinheimo O, et al. Plasma concentrations and receptor binding of RU 486 and its metabolites in humans. J Steroid Biochem. 1987 Feb;26(2):279-84. |