Bioactivity | (d(CH2)51,Tyr(Me)2,Dab5,Arg8)-Vasopressin (d(CH2)5[Tyr(Me)2, Dab5]AVP) is a specific antagonist of vasopressin V1a receptor, with a pA2 of 6.71[1]. |
Name | (d(CH2)51,Tyr(Me)2,Dab5,Arg8)-Vasopressin |
CAS | 176714-12-8 |
Sequence | {Mpa(Cyclohexyl)}-{Tyr(Me)}-Phe-Gln-{Dab}-Cys-Pro-Arg-Gly-NH2 (Disulfide bridge: Mpa1-Cys6) |
Shortening | {Mpa(Cyclohexyl)}-{Tyr(Me)}-FQ-{Dab}-CPRG-NH2 (Disulfide bridge: Mpa1-Cys6) |
Formula | C52H76N14O11S2 |
Molar Mass | 1137.38 |
Transport | Room temperature in continental US; may vary elsewhere. |
Storage | Please store the product under the recommended conditions in the Certificate of Analysis. |
Reference | [1]. Chan WY, et, al. Discovery and design of novel and selective vasopressin and oxytocin agonists and antagonists: the role of bioassays. Exp Physiol. 2000 Mar;85 Spec No:7S-18S. |