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(d(CH2)51,Tyr(Me)2,Arg8)-Vasopressin

CAS: 73168-24-8 F: C52H74N14O12S2 W: 1151.36

(d(CH2)51,Tyr(Me)2,Arg8)-Vasopressin (SKF 100273) is a vasopressin V1 receptor selective antagonist.
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This product is for research use only, not for human use. We do not sell to patients.

Bioactivity (d(CH2)51,Tyr(Me)2,Arg8)-Vasopressin (SKF 100273) is a vasopressin V1 receptor selective antagonist[1].
Name (d(CH2)51,Tyr(Me)2,Arg8)-Vasopressin
CAS 73168-24-8
Sequence {Pmp}-{Tyr(Me)}-Phe-Gln-Asn-Cys-Pro-Arg-Gly-NH2 (Disulfide bond: Pmp1-Cys6) (Pmp=β-Mercapto-β,β-cyclopentamethylene-propionic acid)
Shortening {Pmp}-{Tyr(Me)}-FQNCPRG-NH2 (Disulfide bond: Pmp1-Cys6) (Pmp=β-Mercapto-β,β-cyclopentamethylene-propionic acid)
Formula C52H74N14O12S2
Molar Mass 1151.36
Transport Room temperature in continental US; may vary elsewhere.
Storage

Please store the product under the recommended conditions in the Certificate of Analysis.

Reference [1]. Arai Y, et al. New topics in vasopressin receptors and approach to novel drugs: research and development of conivaptan hydrochloride (YM087), a drug for the treatment of hyponatremia. J Pharmacol Sci. 2009 Jan;109(1):53-9.