Bioactivity | (d(CH2)51,Tyr(Me)2,Arg8)-Vasopressin (SKF 100273) is a vasopressin V1 receptor selective antagonist[1]. |
Name | (d(CH2)51,Tyr(Me)2,Arg8)-Vasopressin |
CAS | 73168-24-8 |
Sequence | {Pmp}-{Tyr(Me)}-Phe-Gln-Asn-Cys-Pro-Arg-Gly-NH2 (Disulfide bond: Pmp1-Cys6) (Pmp=β-Mercapto-β,β-cyclopentamethylene-propionic acid) |
Shortening | {Pmp}-{Tyr(Me)}-FQNCPRG-NH2 (Disulfide bond: Pmp1-Cys6) (Pmp=β-Mercapto-β,β-cyclopentamethylene-propionic acid) |
Formula | C52H74N14O12S2 |
Molar Mass | 1151.36 |
Transport | Room temperature in continental US; may vary elsewhere. |
Storage | Please store the product under the recommended conditions in the Certificate of Analysis. |
Reference | [1]. Arai Y, et al. New topics in vasopressin receptors and approach to novel drugs: research and development of conivaptan hydrochloride (YM087), a drug for the treatment of hyponatremia. J Pharmacol Sci. 2009 Jan;109(1):53-9. |