| Bioactivity | (S,R,S)-AHPC-PEG4-N3 is a synthesized E3 ligase ligand-linker conjugate that incorporates the (S,R,S)-AHPC based VHL ligand and 4-unit PEG linker used in PROTAC technology. | ||||||||||||
| Invitro | E3 ligase Ligand-Linker Conjugates 4 together with JQ1 triggers the intracellular destruction of BET proteins[1]. | ||||||||||||
| Name | (S,R,S)-AHPC-PEG4-N3 | ||||||||||||
| CAS | 1797406-81-5 | ||||||||||||
| Formula | C32H47N7O8S | ||||||||||||
| Molar Mass | 689.82 | ||||||||||||
| Appearance | Viscous liquid | ||||||||||||
| Transport | Room temperature in continental US; may vary elsewhere. | ||||||||||||
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| Reference | [1]. Zengerle M, et al. Selective Small Molecule Induced Degradation of the BET Bromodomain Protein BRD4. ACS Chemical Biology (2015), 10(8), 1770-1777. |
(S,R,S)-AHPC-PEG4-N3
CAS: 1797406-81-5 F: C32H47N7O8S W: 689.82
(S,R,S)-AHPC-PEG4-N3 is a synthesized E3 ligase ligand-linker conjugate that incorporates the (S,R,S)-AHPC based VHL lig
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