Bioactivity | (S)-Sitagliptin phosphate is the less active S-enantiomer of Sitagliptin phosphate. Sitagliptin phosphate (MK-0431 phosphate) is a potent inhibitor of DPP4 with an IC50 of 19 nM in Caco-2 cell extracts[1]. |
Name | (S)-Sitagliptin phosphate |
CAS | 823817-58-9 |
Formula | C16H18F6N5O5P |
Molar Mass | 505.31 |
Transport | Room temperature in continental US; may vary elsewhere. |
Storage | Please store the product under the recommended conditions in the Certificate of Analysis. |
Reference | [1]. Chi-Hung Ho, et al. Biocatalytic Continuous Manufacturing of Diabetes Drug: Plantwide Process Modeling, Optimization, and Environmental and Economic Analysis. ACS Sustainable Chem. Eng. 2019, 7, 1, 1038-1051. |