(R)-ZINC-3573_product_DataBase

CAS: 2089389-15-9 F: C18H21N5 W: 307.39

(R)-ZINC-3573 is a selective Mas-related G protein-coupled receptor X2 (MRGPRX2) agonist with an EC50 value of 740 nM. (

This product is for research use only, not for human use. We do not sell to patients.

Bioactivity

(R)-ZINC-3573 is a selective Mas-related G protein-coupled receptor X2 (MRGPRX2) agonist with an EC50 value of 740 nM. (R)-ZINC-3573 can be used as a MRGPRX2 probe for the research of pain and itch[1].

Invitro

(R)-ZINC-3573 (0.001 nM-100 μM) 促进 β-己糖胺酶脱颗粒并诱导 LAD2 肥大细胞胞内钙释放[1]。

Name

(R)-ZINC-3573

CAS

2089389-15-9

Formula

C18H21N5

Molar Mass

307.39

Appearance

Solid

Transport

Room temperature in continental US; may vary elsewhere.

Storage

Powder	-20°C	3 years
	4°C	2 years
In solvent	-80°C	6 months
	-20°C	1 month

Reference

[1]. Lansu K, et al. In silico design of novel probes for the atypical opioid receptor MRGPRX2. Nat Chem Biol. 2017 May;13(5):529-536.

PeptideDB

(R)-ZINC-3573

CAS: 2089389-15-9 F: C18H21N5 W: 307.39