Bioactivity | (R)-VT104 is the R-enantiomer of VT104. (R)-VT104 shows an IC50 value of 0.1-1 μΜ for firefly luciferase. VT104 is an orally active and pan-TEAD auto-palmitoylation inhibitor[1]. | ||||||||||||
Name | (R)-VT104 | ||||||||||||
CAS | 2417718-26-2 | ||||||||||||
Formula | C25H19F3N2O | ||||||||||||
Molar Mass | 420.43 | ||||||||||||
Appearance | Solid | ||||||||||||
Transport | Room temperature in continental US; may vary elsewhere. | ||||||||||||
Storage |
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Reference | [1]. Konradi, Andrei W, et al. Preparation of substituted naphthalene-2-carboxamide derivatives useful for treatment of cancer. WO2020097389. |