(R)-Simurosertib_product_DataBase

CAS: 1330782-69-8 F: C17H19N5OS W: 341.43

(R)-Simurosertib ((R)-TAK-931) is the (R)-enantiomer of Simurosertib. Simurosertib (TAK-931) is an orally active, select

This product is for research use only, not for human use. We do not sell to patients.

Bioactivity

(R)-Simurosertib ((R)-TAK-931) is the (R)-enantiomer of Simurosertib. Simurosertib (TAK-931) is an orally active, selective and ATP-competitive cell division cycle 7 (CDC7) kinase inhibitor, with an IC50 of <0.3 nM [1].

Name

(R)-Simurosertib

CAS

1330782-69-8

Formula

C17H19N5OS

Molar Mass

341.43

Appearance

Solid

Transport

Room temperature in continental US; may vary elsewhere.

Storage

Powder	-20°C	3 years
	4°C	2 years
In solvent	-80°C	6 months
	-20°C	1 month

Reference

[1]. K Iwai, et al. A novel CDC7-selective inhibitor TAK-931 with potent antitumor activity. European Journal of Cancer , 2016 , 69 (1) :S34.

PeptideDB

(R)-Simurosertib

CAS: 1330782-69-8 F: C17H19N5OS W: 341.43