| Bioactivity | (R)-NVP-CGM097 is the R-enantiomer of NVP-CGM097 (HY-15954). NVP-CGM097 is a potent and selective MDM2 inhibitor with an IC50 of 1.7 nM for hMDM2[1]. |
| CAS | 2643938-26-3 |
| Formula | C38H47ClN4O4 |
| Molar Mass | 659.26 |
| Transport | Room temperature in continental US; may vary elsewhere. |
| Storage | Please store the product under the recommended conditions in the Certificate of Analysis. |
| Reference | [1]. Holzer P, et al. Discovery of a Dihydroisoquinolinone Derivative (NVP-CGM097): A Highly Potent and Selective MDM2 Inhibitor Undergoing Phase 1 Clinical Trials in p53wt Tumors. J Med Chem. 2015 Aug 27;58(16):6348-58. |
(R)-NVP-CGM097
CAS: 2643938-26-3 F: C38H47ClN4O4 W: 659.26
(R)-NVP-CGM097 is the R-enantiomer of NVP-CGM097 (HY-15954). NVP-CGM097 is a potent and selective MDM2 inhibitor with an
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