| Bioactivity | (N-Me-Tyr1,N-Me-Arg7,D-Leu-NHEt8)-Dynorphin A (1-8) (E-2078), a stable Dynorphin A (1–8) (HY-P2159) analog, is a kappa opioid receptor (KOR) agonist[1]. |
| Name | (N-Me-Tyr1,N-Me-Arg7,D-Leu-NHEt8)-Dynorphin A (1-8) |
| CAS | 103613-84-9 |
| Sequence | {Tyr(Me)}-Gly-Gly-Phe-Leu-Arg-{Arg(N-Me)}-{d-Leu}-{NHEt} |
| Shortening | {Tyr(Me)}-GGFLR-{Arg(N-Me)}-{d-Leu}-{NHEt} |
| Formula | C50H81N15O9 |
| Molar Mass | 1036.27 |
| Transport | Room temperature in continental US; may vary elsewhere. |
| Storage | Please store the product under the recommended conditions in the Certificate of Analysis. |
| Reference | [1]. Butelman ER, et al. Effects of E-2078, a stable dynorphin A(1-8) analog, on sedation and serum prolactin levels in rhesus monkeys. Psychopharmacology (Berl). 1999 Nov;147(1):73-80. |