Bioactivity | (D-Arg2, Sar 4)-Dermorphin (1-4) is a tetrapeptide derivative of Dermorphin (HY-P0244) isolated from amphibian skin. (D-Arg2, Sar 4)-Dermorphin (1-4) has a significant analgesic effect by binding to μ-opioid receptors (MOR) in the body. (D-Arg2, Sar 4)-Dermorphin (1-4) can be used in the development of analgesic drugs[1]. |
CAS | 90549-86-3 |
Sequence | Tyr-{DArg}-Phe-{Sar} |
Shortening | Y-{DArg}-F-{Sar} |
Formula | C27H37N7O6 |
Molar Mass | 555.63 |
Transport | Room temperature in continental US; may vary elsewhere. |
Storage | Please store the product under the recommended conditions in the Certificate of Analysis. |
Reference | [1]. Nakata N, et al. Physical dependence of a dermorphin tetrapeptide analog,[D-Arg2, Sar4]-dermorphin (1–4) in the rat[J]. Pharmacology Biochemistry and Behavior, 1986, 24(1): 27-31. |