Bioactivity | (Ala13)-Apelin-13 TFA is a potent apelin receptors (APJ) antagonist. (Ala13)-Apelin-13 TFA inhibits gastric motility through vagal cholinergic pathway[1]. | ||||||
In Vivo | (Ala13)-Apelin-13 TFA (1-300 pmol/60 nl;显微注射到 DVC 中) 以剂量依赖性方式降低大鼠的胃张力和胃动力[1]。 | ||||||
Name | (Ala13)-Apelin-13 TFA | ||||||
Formula | C63H107N23O16S.xC2HF3O2 | ||||||
Molar Mass | 1474.73 (free acid) | ||||||
Appearance | 固体 | ||||||
Transport | Room temperature in continental US; may vary elsewhere. | ||||||
Storage | Sealed storage, away from moisture and light
*In solvent : -80°C, 6 months; -20°C, 1 month (sealed storage, away from moisture and light) |
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Reference | [1]. Bülbül M, et al. Apelin-13 inhibits gastric motility through vagal cholinergic pathway in rats. Am J Physiol Gastrointest Liver Physiol. 2018 Feb 1;314(2):G201-G210. |