(1S,2S)-2-PCCA hydrochloride_product_DataBase

Bioactivity	(1S,2S)-2-PCCA hydrochloride is a less active diastereomer of 2-PCCA. 2-PCCA is a GPR88 receptor agonist, and inhibits GPR88-mediated cAMP production, with an EC50 of 116 nM in HEK293 cells.
Target	GPR88 receptor
Invitro	(1S,2S)-2-PCCA hydrochloride is a less active diastereomer of 2-PCCA. (1R,2R)-2-PCCA is approximately 5-fold more potent than (1S,2S)-2-PCCA[1]. MCE has not independently confirmed the accuracy of these methods. They are for reference only. 0 --> (1S,2S)-2-PCCA hydrochloride 相关抗体:
CAS	1609563-70-3
Formula	C30H39Cl2N3O
Molar Mass	528.56
Appearance	固体
Transport	Room temperature in continental US; may vary elsewhere.
Storage	4°C, stored under nitrogen *In solvent : -80°C, 6 months; -20°C, 1 month (stored under nitrogen)
Reference	[1]. Jin C, et al. Synthesis, pharmacological characterization, and structure-activity relationship studies of small molecular agonists for the orphan GPR88 receptor. ACS Chem Neurosci. 2014 Jul 16;5(7):576-87.

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