| Description | PTGR2-IN-1 is a potent inhibito of PTGR2r(IC50 : 0.7 μM). It increases 15-keto-PGE2-dependent PPARγ transcriptional activity in PTGR2-transfected HEK293T cells. |
| Target activity | PTGR2:0.7 μM |
| Synonyms | PTGR2-IN-22 |
| molecular weight | 310.39 |
| Molecular formula | C19H22N2O2 |
| CAS | 349093-44-3 |
| Storage | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice. |
| Solubility | DMSO: 100 mg/mL (322.18 mM), Sonication is recommended. |
| References | 1. Parker CG, et al. Ligand and Target Discovery by Fragment-Based Screening in Human Cells. Cell. 2017;168(3):527-541.e29. |