| Description | PKC-theta inhibitor is PKC-θinhibitor, with an IC50 of 12 nM. |
| Target activity | PKCθ:12 nM |
| molecular weight | 454.45 |
| Molecular formula | C20H25F3N6O3 |
| CAS | 736048-65-0 |
| Storage | Powder: -20°C for 3 years | In solvent: -80°C for 1 year |
| Solubility | DMSO: 62.5 mg/mL (137.53 mM) |
| References | 1. Cywin CL, et al. Discovery of potent and selective PKC-theta inhibitors. Bioorg Med Chem Lett. 2007 Jan 1;17(1):225-30. |