| Description | PKC-theta inhibitor hcl is a selective PKC-θinhibitor(IC50:12 nM). |
| Target activity | PKCθ:12 nM |
| Synonyms | PKC-theta inhibitor |
| molecular weight | 490.91 |
| Molecular formula | C20H26ClF3N6O3 |
| CAS | 2253640-49-0 |
| Storage | Powder: -20°C for 3 years | In solvent: -80°C for 1 year |
| Solubility | DMSO: 55 mg/mL (121.04 mM), Sonication is recommended. |
| References | 1. Cywin C L , Dahmann G , Iii A S P , et al. Discovery of potent and selective PKC-θ inhibitors[J]. Bioorganic & Medicinal Chemistry Letters, 2007, 17(1):225-230. |