| Description | LDN-27219 is a potent hTGase inhibitor with IC50 of 0.6 uM. |
| Target activity | TGase (human):0.6 uM |
| molecular weight | 408.5 |
| Molecular formula | C20H16N4O2S2 |
| CAS | 312946-37-5 |
| Storage | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice. |
| Solubility | DMSO: 100 mg/mL (244.8 mM), Sonication is recommended. |
| References | 1. Case A, et al. Kinetic analysis of the interaction of tissue transglutaminase with a nonpeptidic slow-binding inhibitor. Biochemistry. 2007 Jan 30;46(4):1106-15. |