| Description | HPP-9, a Proteolysis-Targeting Chimera (PROTAC) derived from Hedgehog Pathway Inhibitor-1 (HPI-1) with a pIC50 value of 6.71, is designed to degrade BET bromodomains and exhibits antitumor activity [1]. |
| molecular weight | 900.97 |
| Molecular formula | C49H52N6O11 |
| Storage | Powder: -20°C for 3 years | In solvent: -80°C for 1 year |