| Description | CPFPX is a highly selective radioactive ligand for the A1 adenosine receptor (A1AR). |
| Synonyms | [18F]CPFPX |
| molecular weight | 321.38 |
| Molecular formula | C16H23FN4O2 |
| CAS | 227205-79-0 |
| Storage | Powder: -20°C for 3 years | In solvent: -80°C for 1 year |
| References | 1. Kroll T, Elmenhorst D, Weisshaupt A, Beer S, Bauer A. Reproducibility of non-invasive a1 adenosine receptor quantification in the rat brain using [(18)F]CPFPX and positron emission tomography. Mol Imaging Biol. 2014 Oct;16(5):699-709. doi: 10.1007/s11307-014-0729-0. PubMed PMID: 24595700. 2. Elmenhorst D, Kroll T, Wedekind F, Weisshaupt A, Beer S, Bauer A. In vivo kinetic and steady-state quantification of 18F-CPFPX binding to rat cerebral A1 adenosine receptors: validation by displacement and autoradiographic experiments. J Nucl Med. 2013 Aug;54(8):1411-9. doi: 10.2967/jnumed.112.115576. PubMed PMID: 23740103. 3. Elmenhorst D, Meyer PT, Matusch A, Winz OH, Bauer A. Caffeine occupancy of human cerebral A1 adenosine receptors: in vivo quantification with 18F-CPFPX and PET. J Nucl Med. 2012 Nov;53(11):1723-9. doi: 10.2967/jnumed.112.105114. PubMed PMID: 22966134. |