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Contezolid acefosamil

CAS No.: 1807497-11-5

Contezolid acefosamil (MRX-4), an orally active prodrug, is metabolized into Contezolid (MRX-I), an oxazolidinone deriva
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Description Contezolid acefosamil (MRX-4), an orally active prodrug, is metabolized into Contezolid (MRX-I), an oxazolidinone derivative with potent in vitro efficacy against multidrug-resistant Gram-positive bacteria, including MRSA.
Synonyms MRX-4, Contezolid acefosamil
molecular weight 530.353
Molecular formula C20H18F3N4O8P
CAS 1807497-11-5
Storage Powder: -20°C for 3 years | In solvent: -80°C for 1 year
References 1. Matteo Bassetti, et al. Innovative therapies for acute bacterial skin and skin-structure infections (ABSSSI) caused by methicillin-resistant Staphylococcus aureus: advances in phase I and II trials. Expert Opin Investig Drugs. 2020 May;29(5):495-506.