| Description | BMS-505130 is an effective selective serotonin transport inhibitor. |
| Synonyms | UNII-E892TW82D9, E892TW82D9, BMS-505130 free base |
| molecular weight | 355.39 |
| Molecular formula | C19H21N3O4 |
| CAS | 859230-84-5 |
| Storage | Powder: -20°C for 3 years | In solvent: -80°C for 1 year |
| References | 1. Mattson RJ, Catt JD, Denhart DJ, Deskus JA, Ditta JL, Higgins MA, Marcin LR, Sloan CP, Beno BR, Gao Q, Cunningham MA, Mattson GK, Molski TF, Taber MT, Lodge NJ. Conformationally restricted homotryptamines. 2. Indole cyclopropylmethylamines as selective serotonin reuptake inhibitors. J Med Chem. 2005 Sep 22;48(19):6023-34. PubMed PMID: 16162005. 2. Marcin LR, Denhart DJ, Mattson RJ. Catalytic asymmetric diazoacetate cyclopropanation of 1-tosyl-3-vinylindoles. A route to conformationally restricted homotryptamines. Org Lett. 2005 Jun 23;7(13):2651-4. PubMed PMID: 15957913. 3. Taber MT, Wright RN, Molski TF, Clarke WJ, Brassil PJ, Denhart DJ, Mattson RJ, Lodge NJ. Neurochemical, pharmacokinetic, and behavioral effects of the novel selective serotonin reuptake inhibitor BMS-505130. Pharmacol Biochem Behav. 2005 Mar;80(3):521-8. PubMed PMID: 15740795. |