| CAS | 500170-27-4 |
| Sequence | 3-Mercaptopropionyl-Tyr-Phe-β-cyclohexyl-Ala-Asn-Cys-Pro-Arg-Gly-NH2 (Disulfide bond) |
| Sequence Single | 3-Mercaptopropionyl-YF-β-cyclohexyl-ANCPRG-NH2 |
| Molecular Formula | C50H71N13O11S2 |
| Molecular Weight | 1094.33 |
| Synonyms | (Deamino-Cys1,Cha4,Arg8)-Vasopressin |
| Technology | Synthetic |
| Storage | -20°C, avoid light, cool and dry place |
| Description | (Deamino-Cys1,β-cyclohexyl-Ala4,Arg8)-Vasopressin also called (Deamino-Cys1,Cha4,Arg8)-Vasopressin, is a potent and selective vasopressin (AVP) V1b receptor agonist with a Ki of 1.2 nM for human V1b receptor. (Deamino-Cys1,β-cyclohexyl-Ala4,Arg8)-Vasopressin shows more selective for V1b receptor than human V1a receptor, V2 receptor, and oxytocin receptors. |
| References | 1. Design of potent and selective agonists for the human vasopressin V1b receptor based on modifications of [deamino-cys1]arginine vasopressin at position 4. Ling Ling Cheng, et al. J Med Chem. 2004 Apr 22;47(9):2375-88. 2. Selectivity of d[Cha4]AVP and SSR149415 at human vasopressin and oxytocin receptors: evidence that SSR149415 is a mixed vasopressin V1b/oxytocin receptor antagonist. Cristiana Griffante, et al. Br J Pharmacol. 2005 Nov;146(5):744-51. |
(Deamino-Cys1,β-cyclohexyl-Ala4,Arg8)-Vasopressin
CAS No.: 500170-27-4
(Deamino-Cys1,β-cyclohexyl-Ala4,Arg8)-Vasopressin also called (Deamino-Cys1,Cha4,Arg8)-Vasopressin, is a potent and sel
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