Gumelutamide (monosuccinate) is an androgen antagonist. Gumelutamide (monosuccinate) is a tetrahydropyrido-pyrimidine compound that acts as an antineoplastic agent.

Physicochemical Properties

Molecular Formula	C26H27CLN6O5
Molecular Weight	538.98
CAS #	2842844-51-1
Related CAS #	Gumelutamide monosuccinate;2842844-51-1
Storage	Powder-20°C 3 years 4°C 2 years In solvent -80°C 6 months -20°C 1 month
Shipping Condition	Room temperature (This product is stable at ambient temperature for a few days during ordinary shipping and time spent in Customs)

Biological Activity

References

[1]. Preparation of novel tetrahydropyridopyrimidine compounds, and antiandrogens and antitumor agents containing them: World Intellectual Property Organization, WO2015182712. 2015-12-03. [2]. WHO Drug Information-World Health Organization (WHO).

Solubility Data

Preparing Stock Solutions		1 mg	5 mg	10 mg
	1 mM	1.8554 mL	9.2768 mL	18.5536 mL
	5 mM	0.3711 mL	1.8554 mL	3.7107 mL
	10 mM	0.1855 mL	0.9277 mL	1.8554 mL

*Note: Please select an appropriate solvent for the preparation of stock solution based on your experiment needs. For most products, DMSO can be used for preparing stock solutions (e.g. 5 mM, 10 mM, or 20 mM concentration); some products with high aqueous solubility may be dissolved in water directly. Solubility information is available at the above Solubility Data section. Once the stock solution is prepared, aliquot it to routine usage volumes and store at -20°C or -80°C. Avoid repeated freeze and thaw cycles.